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Functionalization of the imidazo[1,2-a]pyridine ring in ?-phosphonoacrylates and ?-phosphonopropionates via microwave-assisted Mizoroki-Heck reaction.

ABSTRACT: A series of new phosphonocarboxylates containing an imidazo[1,2-a]pyridine ring has been synthesized via the microwave-assisted Mizoroki-Heck reaction. The efficient modification of the imidazo[1,2-a]pyridine ring has been achieved as late-stage functionalization, enabling and accelerating the generation of a library of compounds from a common precursor.

SUBMITTER: Kusy D 

PROVIDER: S-EPMC6964661 | biostudies-literature | 2020

REPOSITORIES: biostudies-literature

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Functionalization of the imidazo[1,2-<i>a</i>]pyridine ring in α-phosphonoacrylates and α-phosphonopropionates via microwave-assisted Mizoroki-Heck reaction.

Kusy Damian D   Wojciechowska Agata A   Małolepsza Joanna J   Błażewska Katarzyna M KM  

Beilstein journal of organic chemistry 20200103

A series of new phosphonocarboxylates containing an imidazo[1,2-<i>a</i>]pyridine ring has been synthesized via the microwave-assisted Mizoroki-Heck reaction. The efficient modification of the imidazo[1,2-<i>a</i>]pyridine ring has been achieved as late-stage functionalization, enabling and accelerating the generation of a library of compounds from a common precursor. ...[more]

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