Disrupting enzyme fluidity.
Ontology highlight
ABSTRACT:
SUBMITTER: Anand GS
PROVIDER: S-EPMC7834015 | biostudies-literature | 2021 Jan
REPOSITORIES: biostudies-literature
Publications
A combination of X-ray crystallography, NMR, and mass spectrometry has revealed how diverse small-molecule inhibitors bind Bruton's tyrosine kinase and alter the conformation of this enzyme. ...[more]
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